Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-[2-[4-[(dimethylamino)methyl]phenyl]ethyl]-7-[(4-fluorophenyl)methyl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1-one
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 PubChem ID
CID: 155562407
Canonical SMILES
CN(C)Cc1ccc(CCN2CCn3cc(Cc4ccc(F)cc4)cc3C2=O)cc1
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Compound Formula C25H28FN3O
Compound Structure
Protein Name
 Protein Info 
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 228 nM
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