Brief Information of the Compound and Protein
Compound Name
(R)-4-((1-(benzo[d][1,3]dioxol-5-ylmethyl)piperidin-4-yl)methyl)-N-(1-(4-bromophenyl)ethyl)benzamide
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PubChem ID
CID: 12020151
Canonical SMILES
C[C@@H](NC(=O)c1ccc(CC2CCN(Cc3ccc4OCOc4c3)CC2)cc1)c1ccc(Br)cc1
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Compound Formula C29H31BrN2O3
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 101 nM