Brief Information of the Compound and Protein
Compound Name
3-amino-4-methyl-7-oxo-N-[[4-(trifluoromethylsulfonyl)phenyl]methyl]-6H-thieno[2,3-c]pyridine-2-carboxamide
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PubChem ID
CID: 75203027
Canonical SMILES
Cc1c[nH]c(=O)c2sc(C(=O)NCc3ccc(cc3)S(=O)(=O)C(F)(F)F)c(N)c12
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Compound Formula C17H14F3N3O4S2
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 260 nM
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