Brief Information of the Compound and Protein
Compound Name
1-[5-[(3R)-3-[6-(cyclopropylmethoxy)pyridin-3-yl]oxy-2-oxopyrrolidin-1-yl]pyrimidin-2-yl]azetidine-3-carboxylic acid
    Show/Hide
PubChem ID
CID: 139437014
Canonical SMILES
OC(=O)C1CN(C1)c1ncc(cn1)N1CC[C@@H](Oc2ccc(OCC3CC3)nc2)C1=O
    Show/Hide
Compound Formula C21H23N5O5
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 4920 nM
   TI
   LI
   LO
   TS