Brief Information of the Compound and Protein
| Compound Name |
(1R)-8-chloro-2,3,4,5-tetrahydro-1-methyl-1H-3-benzazepine
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
5-hydroxytryptamine receptor 2B
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Protein Classification |
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
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| Uniprot ID | Gene Name | HTR2B |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Biochemical Assays
| 1 | Ki = 1.3 nM | ||
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| 2 | Ki = 174 nM | ||
| 3 | Ki = 189 nM | ||
| 4 | Ki = 220 nM | ||