Brief Information of the Compound and Protein
| Compound Name |
Faridak
Show/Hide
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
Histone deacetylase 5
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Protein Classification |
Epigenetic regulator
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Eraser
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Histone deacetylase
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HDAC class IIa
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| Uniprot ID | Gene Name | HDAC5 |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
| Cell Line ID | Cell Line Name | Cell Line Organism | |
| CL000013 | Sf9 | Spodoptera frugiperda (Fall armyworm) | 3 |
| 1 |
IC50 = 92 nM
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TI
LI
LO
TS
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|---|---|---|---|
| 2 |
IC50 = 190.3 nM
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TI
LI
LO
TS
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| 3 |
IC50 > 20000 nM
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TI
LI
LO
TS
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Biochemical Assays
| 1 | IC50 = 7.8 nM | ||
|---|---|---|---|
| 2 | IC50 = 190 nM | ||
| 3 | IC50 = 195.6 nM | ||
| 4 | IC50 = 290 nM | ||
| 5 | IC50 < 300 nM | ||
| 6 | Ki = 0.7 nM | ||
| 7 | Ki = 57 nM | ||
| 8 | Ki = 80 nM | ||