Brief Information of the Compound and Protein
Compound Name
4-[4-(3-methoxypyridin-2-yl)piperidin-1-yl]-1-pyrazin-2-ylazepane
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PubChem ID
CID: 155524827
Canonical SMILES
COc1cccnc1C1CCN(CC1)C1CCCN(CC1)c1cnccn1
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Compound Formula C21H29N5O
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08172
Gene Name
CHRM2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 250 nM
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