Brief Information of the Compound and Protein
Compound Name
2-[(1S,5R)-6-(1-phenylimidazol-2-yl)-3-azabicyclo[3.1.0]hexan-3-yl]-6-pyrazin-2-yl-6-azaspiro[3.4]octane
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Canonical SMILES
C1C(CC11CCN(C1)c1cnccn1)N1C[C@H]2[C@@H](C1)[C@H]2c1nccn1-c1ccccc1
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Compound Formula C25H28N6
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08172
Gene Name
CHRM2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 420 nM
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