Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(E)-N1-(3-Methoxyphenyl)-N3-(3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)malonamide
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 PubChem ID
CID: 141764130
Canonical SMILES
COc1cccc(NC(=O)CC(=O)Nc2ccc3c(/C=C/c4ccccn4)n[nH]c3c2)c1
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Compound Formula C24H21N5O3
Compound Structure
Protein Name
 Protein Info 
Mast/stem cell growth factor receptor Kit
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
TK protein kinase group
>
Tyrosine protein kinase PDGFR family
Uniprot ID
P10721
Gene Name
KIT
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3
 Cell Line Info 
Mus musculus (Mouse)  2
1
GI50 = 234 nM
   TI
   LI
   LO
   TS
2
GI50 = 2740 nM
   TI
   LI
   LO
   TS