Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-[(1S)-1-(2,3-dichloro-4-pyrazin-2-ylphenyl)ethyl]-2-[(1R)-5-(6-methylpyrimidin-4-yl)-2,3-dihydro-1H-inden-1-yl]-2,7-diazaspiro[3.5]nonane-7-carboxamide
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 PubChem ID
CID: 145981196
Canonical SMILES
C[C@H](NC(=O)N1CCC2(CN(C2)[C@@H]2CCc3cc(ccc23)-c2cc(C)ncn2)CC1)c1ccc(-c2cnccn2)c(Cl)c1Cl
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Compound Formula C34H35Cl2N7O
Compound Structure
Protein Name
 Protein Info 
Growth hormone secretagogue receptor type 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
Q92847
Gene Name
GHSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  3
1
EC50 = 483 nM
   TI
   LI
   LO
   TS
2
EC50 > 30000 nM
   TI
   LI
   LO
   TS
3
IC50 = 1210 nM
   TI
   LI
   LO
   TS