Brief Information of the Compound and Protein
Compound Name
N-[(3R,4S)-3-hydroxyoxan-4-yl]-4-[[4-(4-hydroxypyrazol-1-yl)phenyl]methyl]-5-methylpyridine-2-carboxamide
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PubChem ID
CID: 145969027
Canonical SMILES
Cc1cnc(cc1Cc1ccc(cc1)-n1cc(O)cn1)C(=O)N[C@H]1CCOC[C@@H]1O
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Compound Formula C22H24N4O4
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P11229
Gene Name
CHRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 70 nM
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