Brief Information of the Compound and Protein
Compound Name
N-[(1S,2S)-2-hydroxycyclohexyl]-6-(hydroxymethyl)-1-methyl-2-oxo-5-[(4-pyrazol-1-ylphenyl)methyl]pyridine-3-carboxamide
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PubChem ID
CID: 145969714
Canonical SMILES
Cn1c(CO)c(Cc2ccc(cc2)-n2cccn2)cc(C(=O)N[C@H]2CCCC[C@@H]2O)c1=O
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Compound Formula C24H28N4O4
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P11229
Gene Name
CHRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 40 nM
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