Brief Information of the Compound and Protein
Compound Name
5-methyl-4-[(4-pyrazol-1-ylphenyl)methyl]-N-[(2R,3S)-1,2,5-trihydroxypentan-3-yl]pyridine-2-carboxamide
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PubChem ID
CID: 145969071
Canonical SMILES
Cc1cnc(cc1Cc1ccc(cc1)-n1cccn1)C(=O)N[C@@H](CCO)[C@@H](O)CO
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Compound Formula C22H26N4O4
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P11229
Gene Name
CHRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 > 300 nM
   TI
   LI
   LO
   TS