Brief Information of the Compound and Protein
Compound Name
1-[9-chloro-1-(2,4-dichlorophenyl)-3,4-dihydro-2H-pyrimido[1,2-a]benzimidazol-6-yl]propan-1-one
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PubChem ID
CID: 57786300
Canonical SMILES
CCC(=O)c1ccc(Cl)c2nc3N(CCCn3c12)c1ccc(Cl)cc1Cl
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Compound Formula C19H16Cl3N3O
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 210 nM
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