Brief Information of the Compound and Protein
Compound Name
[2-chloro-4-(3-methylpyrazol-1-yl)phenyl]-[5-(dimethylamino)-2,3,4,5-tetrahydro-1-benzazepin-1-yl]methanone
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PubChem ID
CID: 145966126
Canonical SMILES
CN(C)C1CCCN(C(=O)c2ccc(cc2Cl)-n2ccc(C)n2)c2ccccc12
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Compound Formula C23H25ClN4O
Compound Structure
Protein Name
Vasopressin V2 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Vasopressin and oxytocin receptor
Uniprot ID
P30518
Gene Name
AVPR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 331 nM
   TI
   LI
   LO
   TS