Brief Information of the Compound and Protein
Compound Name
4-[(2R,3R)-3-(3,5-dichlorophenyl)-6,6-dimethylmorpholin-2-yl]oxy-2,5-difluoro-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide
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PubChem ID
CID: 145969142
Canonical SMILES
CC1(C)CN[C@@H]([C@@H](Oc2cc(F)c(cc2F)S(=O)(=O)Nc2ncns2)O1)c1cc(Cl)cc(Cl)c1
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Compound Formula C20H18Cl2F2N4O4S2
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 6000 nM
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