Brief Information of the Compound and Protein
Compound Name
N-[[5-tert-butyl-2-[4-[(E)-2-(4-methylphenyl)ethenyl]phenyl]pyrazol-3-yl]methyl]-2-[3-fluoro-4-(methanesulfonamido)phenyl]propanamide
    Show/Hide
PubChem ID
CID: 145965659
Canonical SMILES
CC(C(=O)NCc1cc(nn1-c1ccc(\C=C\c2ccc(C)cc2)cc1)C(C)(C)C)c1ccc(NS(C)(=O)=O)c(F)c1
    Show/Hide
Compound Formula C33H37FN4O3S
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 819 nM
   TI
   LI
   LO
   TS