Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-Bromo-5-(3-chloro-5-fluorophenoxy)-2,2-difluoro- 3-hydroxy-2,3-dihydrobenzo[b]thiophene 1,1-dioxide
    Show/Hide
 PubChem ID
CID: 118183648
Canonical SMILES
OC1c2c(ccc(Oc3cc(F)cc(Cl)c3)c2Br)S(=O)(=O)C1(F)F
    Show/Hide
Compound Formula C14H7BrClF3O4S
Compound Structure
Protein Name
 Protein Info 
Endothelial PAS domain-containing protein 1
Protein Classification
Transcription factor
Uniprot ID
Q99814
Gene Name
EPAS1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000244 786-O
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 43 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 < 5 nM