Brief Information of the Compound and Protein
Compound Name
3-[4-[5-chloro-6-(2-methylpropoxy)pyridin-3-yl]-2,5-difluorophenyl]-N-cyclopropyl-1H-1,2,4-triazole-5-sulfonamide
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PubChem ID
CID: 145963182
Canonical SMILES
CC(C)COc1ncc(cc1Cl)-c1cc(F)c(cc1F)-c1nnc([nH]1)S(=O)(=O)NC1CC1
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Compound Formula C20H20ClF2N5O3S
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 7300 nM
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