Brief Information of the Compound and Protein
Compound Name
 Compound Info 
1-[3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-(1-methylpiperidin-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone
    Show/Hide
 PubChem ID
CID: 121372830
Canonical SMILES
CN1CCC(CC1)n1nc(N2CCCc3cc(-c4cnn(C)c4)c(cc23)C(F)F)c2CN(CCc12)C(C)=O
    Show/Hide
Compound Formula C28H35F2N7O
Compound Structure
Protein Name
 Protein Info 
CREB-binding protein
Protein Classification
Epigenetic regulator
>
Reader
>
Bromodomain
Uniprot ID
Q92793
Gene Name
CREBBP
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 98 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 2 nM