Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamide
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 PubChem ID
CID: 121372947
Canonical SMILES
Cn1cc(cn1)-c1cc2CCCN(c3nn(C4CCOCC4)c4CCN(Cc34)C(N)=O)c2cc1C(F)F
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Compound Formula C26H31F2N7O2
Compound Structure
Protein Name
 Protein Info 
CREB-binding protein
Protein Classification
Epigenetic regulator
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Bromodomain
Uniprot ID
Q92793
Gene Name
CREBBP
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 28 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 1 nM