Brief Information of the Compound and Protein
Compound Name
N-(2-fluoro-4-methylsulfonylphenyl)-3-[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-d]pyrimidin-7-amine
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PubChem ID
CID: 137647821
Canonical SMILES
CCCc1cnc(nc1)N1CCC(CC1)n1nnc2c(Nc3ccc(cc3F)S(C)(=O)=O)ncnc12
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Compound Formula C23H26FN9O2S
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 82 nM
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