Brief Information of the Compound and Protein
Compound Name
N-(12-chloro-23-methyl-22-oxo-8,19-dioxa-6,23-diazatetracyclo[18.4.0.02,7.09,14]tetracosa-1(24),2(7),3,5,9(14),10,12,20-octaen-4-yl)ethanesulfonamide
    Show/Hide
PubChem ID
CID: 118137846
Canonical SMILES
CCS(=O)(=O)Nc1cnc2Oc3ccc(Cl)cc3CCCCOc3cc(=O)n(C)cc3-c2c1
    Show/Hide
Compound Formula C23H24ClN3O5S
Compound Structure
Protein Name
Bromodomain-containing protein 4
Protein Classification
Epigenetic regulator
>
Reader
>
Bromodomain
Uniprot ID
O60885
Gene Name
BRD4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000095 NCI-H1299 Homo sapiens (Human)  1
1
EC50 = 9.3 nM
   TI
   LI
   LO
   TS