Brief Information of the Compound and Protein
Compound Name
4-ethylsulfonyl-22-methyl-8,18-dioxa-22-azatetracyclo[17.4.0.02,7.09,14]tricosa-1(23),2(7),3,5,9,11,13,19-octaen-21-one
    Show/Hide
PubChem ID
CID: 118137861
Canonical SMILES
CCS(=O)(=O)c1ccc2Oc3ccccc3CCCOc3cc(=O)n(C)cc3-c2c1
    Show/Hide
Compound Formula C23H23NO5S
Compound Structure
Protein Name
Bromodomain-containing protein 4
Protein Classification
Epigenetic regulator
>
Reader
>
Bromodomain
Uniprot ID
O60885
Gene Name
BRD4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000095 NCI-H1299 Homo sapiens (Human)  1
1
EC50 = 26 nM
   TI
   LI
   LO
   TS