Brief Information of the Compound and Protein
Compound Name
4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(pyridin-2-ylmethoxy)-phenylamino]-3-cyano-7-ethoxy-quinolin-6-yl}-amide
    Show/Hide
PubChem ID
CID: 9915743
SID: 14886227
Canonical SMILES
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C
    Show/Hide
Compound Formula C30H29ClN6O3
Compound Structure
Protein Name
Insulin receptor
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
TK protein kinase group
>
Tyrosine protein kinase InsR family
Uniprot ID
P06213
Gene Name
INSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
GI50 = 290 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Kd = 3000 nM