Brief Information of the Compound and Protein
Compound Name
5-chloro-2-fluoro-4-[[(2R,3R)-2-phenyloxan-3-yl]methylamino]-N-(1,3-thiazol-2-yl)benzenesulfonamide
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PubChem ID
CID: 137640507
Canonical SMILES
Fc1cc(NC[C@H]2CCCO[C@H]2c2ccccc2)c(Cl)cc1S(=O)(=O)Nc1nccs1
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Compound Formula C21H21ClFN3O3S2
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 1300 nM
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