Brief Information of the Compound and Protein
Compound Name
4-[[(3aS,7aR)-2,3,4,5,6,7a-hexahydrofuro[2,3-b]pyran-3a-yl]methylamino]-5-chloro-2-fluoro-N-(1,3-thiazol-2-yl)benzenesulfonamide
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PubChem ID
CID: 137638686
Canonical SMILES
Fc1cc(NC[C@]23CCO[C@H]2OCCC3)c(Cl)cc1S(=O)(=O)Nc1nccs1
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Compound Formula C17H19ClFN3O4S2
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 12800 nM
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