Brief Information of the Compound and Protein
Compound Name
(NE)-N-[6-[(1-pyrimidin-4-ylpiperidin-4-yl)amino]-2-thieno[3,2-c]pyridin-6-ylchromen-4-ylidene]hydroxylamine
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PubChem ID
CID: 137635028
Canonical SMILES
O\N=c1/cc(oc2ccc(NC3CCN(CC3)c3ccncn3)cc12)-c1cc2sccc2cn1
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Compound Formula C25H22N6O2S
Compound Structure
Protein Name
Metabotropic glutamate receptor 4
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
Q14833
Gene Name
GRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 53 nM
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