Brief Information of the Compound and Protein
Compound Name
CHEMBL4060400
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Canonical SMILES
Cc1nn2c(O)cc(nc2c1-c1ccc(F)cc1)C1CCN(CC1)C(=O)OCc1ccccc1
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Compound Formula C26H25FN4O3
Compound Structure
Protein Name
Short transient receptor potential channel 6
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q61143
Gene Name
TRPC6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 3240 nM
   TI
   LI
   LO
   TS
2
EC50 = 3910 nM
   TI
   LI
   LO
   TS