Brief Information of the Compound and Protein
Compound Name
CHEMBL4085233
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Canonical SMILES
CCOC(=O)N1CCC(CC1)c1cc(O)n2nc(C)c(-c3ccc(cc3)C(F)(F)F)c2n1
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Compound Formula C22H23F3N4O3
Compound Structure
Protein Name
Short transient receptor potential channel 6
Protein Classification
Ion channel
>
Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q61143
Gene Name
TRPC6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 890 nM
   TI
   LI
   LO
   TS
2
EC50 = 1385 nM
   TI
   LI
   LO
   TS