Brief Information of the Compound and Protein
Compound Name
5-[1-(6-bromopyridine-3-carbonyl)piperidin-4-yl]-3-(4-fluorophenyl)-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
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Canonical SMILES
Cc1nn2c(O)cc(nc2c1-c1ccc(F)cc1)C1CCN(CC1)C(=O)c1ccc(Br)nc1
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Compound Formula C24H21BrFN5O2
Compound Structure
Protein Name
Short transient receptor potential channel 6
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q61143
Gene Name
TRPC6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 12300 nM
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