Brief Information of the Compound and Protein
Compound Name
3-(4-fluorophenyl)-2-methyl-5-(1-propanoylpiperidin-4-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
    Show/Hide
Canonical SMILES
CCC(=O)N1CCC(CC1)c1cc(O)n2nc(C)c(-c3ccc(F)cc3)c2n1
    Show/Hide
Compound Formula C21H23FN4O2
Compound Structure
Protein Name
Short transient receptor potential channel 6
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Transient receptor potential channel
Uniprot ID
Q61143
Gene Name
TRPC6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 28800 nM
   TI
   LI
   LO
   TS