Brief Information of the Compound and Protein
Compound Name
benzyl 4-[3-(4-chlorophenyl)-2-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]piperidine-1-carboxylate
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Canonical SMILES
Cc1nn2c(O)cc(nc2c1-c1ccc(Cl)cc1)C1CCN(CC1)C(=O)OCc1ccccc1
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Compound Formula C26H25ClN4O3
Compound Structure
Protein Name
Short transient receptor potential channel 6
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q61143
Gene Name
TRPC6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 2050 nM
   TI
   LI
   LO
   TS
2
EC50 = 7790 nM
   TI
   LI
   LO
   TS