Brief Information of the Compound and Protein
| Compound Name |
2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
Cytochrome P450 1A1
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Protein Classification |
Enzyme
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Cytochrome P450
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Cytochrome P450 family 1
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Cytochrome P450 family 1A
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Cytochrome P450 1A1
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| Uniprot ID | Gene Name | CYP1A1 |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
| Cell Line ID | Cell Line Name | Cell Line Organism | |
| CL000006 | HEK293 | Homo sapiens (Human) | 3 |
| 1 |
EC50 = 1800 nM
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TI
LI
LO
TS
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|---|---|---|---|
| 2 |
IC50 = 380 nM
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TI
LI
LO
TS
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| 3 |
IC50 > 10000 nM
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TI
LI
LO
TS
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Biochemical Assays
| 1 | IC50 = 11.9 nM | ||
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| 2 | IC50 = 18 nM | ||
| 3 | IC50 = 43 nM | ||
| 4 | IC50 = 53.8 nM | ||
| 5 | IC50 = 60 nM | ||
| 6 | IC50 = 80.3 nM | ||
| 7 | IC50 = 2700 nM | ||