Brief Information of the Compound and Protein
Compound Name
7-bromo-2-N-(4-chloro-2-methoxy-6-methylphenyl)-4-N-ethyl-3-methyl-4-N-(3,3,3-trifluoropropyl)benzimidazole-2,4-diamine
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PubChem ID
CID: 137640280
Canonical SMILES
CCN(CCC(F)(F)F)c1ccc(Br)c2nc(Nc3c(C)cc(Cl)cc3OC)n(C)c12
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Compound Formula C21H23BrClF3N4O
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 18 nM
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