Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(4aR,5aS,8aR,13aS,15E,15aR,15bR)-15-methoxyimino-2,4a,5,5a,7,8,13a,15a,15b,16-decahydro4,6-methanoindolo[3,2,1-ij]oxepino[2,3,4-de]pyrrolo[2,3-h]quinolin-14-one
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 PubChem ID
CID: 137656578
Canonical SMILES
CO\N=C1/[C@@H]2OCC=C3CN4CC[C@@]56[C@@H]4C[C@@H]3[C@@H]2[C@@H]5N(c2ccccc62)C1=O
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Compound Formula C22H23N3O3
Compound Structure
Protein Name
 Protein Info 
Glycine receptor subunit alpha-1
Protein Classification
Ion channel
>
Ligand-gated ion channel
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Glycine receptor
Uniprot ID
P23415
Gene Name
GLRA1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  2
1
IC50 = 75 nM
   TI
   LI
   LO
   TS
2
Ki = 189 nM
   TI
   LI
   LO
   TS