Brief Information of the Compound and Protein
Compound Name
1-(azetidin-1-yl)-2-[4-[2-[(1S,2R)-2-[1-(5-chloropyrimidin-2-yl)piperidin-4-yl]cyclopropyl]ethoxy]-3-fluorophenyl]ethanone
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PubChem ID
CID: 117684497
Canonical SMILES
Fc1cc(CC(=O)N2CCC2)ccc1OCC[C@@H]1C[C@@H]1C1CCN(CC1)c1ncc(Cl)cn1
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Compound Formula C25H30ClFN4O2
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 2.2 nM
   TI
   LI
   LO
   TS