Brief Information of the Compound and Protein
Compound Name
US9199981, F160
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PubChem ID
CID: 71280722
Canonical SMILES
Cc1ccc(-c2noc(n2)C2CC(F)(F)C2)c(C)c1NC(=O)c1cnc2ccccn12
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Compound Formula C22H19F2N5O2
Compound Structure
Protein Name
Mast/stem cell growth factor receptor Kit
Protein Classification
Enzyme
>
Kinase
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Protein Kinase
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TK protein kinase group
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Tyrosine protein kinase PDGFR family
Uniprot ID
P10721
Gene Name
KIT
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000138 M-07e Homo sapiens (Human)  1
1
IC50 = 293 nM
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