Brief Information of the Compound and Protein
Compound Name
 Compound Info 
US9163015, 35
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 PubChem ID
CID: 53373876
SID: 125295574
Canonical SMILES
CN1C(=O)N(c2ccc(Nc3n[nH]c4cccnc34)cc2Cl)C(=O)C1C(C)(C)C
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Compound Formula C20H21ClN6O2
Compound Structure
Protein Name
 Protein Info 
Metabotropic glutamate receptor 4
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
Q14833
Gene Name
GRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 753 nM
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