Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(6S,9R,12R)-6-cyclopropyl-20-fluoro-12-[(4-fluorophenyl)methyl]-8,9-dimethyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(18),19,21-triene-7,10,13-trione
    Show/Hide
 PubChem ID
CID: 56925345
SID: 135607543
Canonical SMILES
C[C@H]1N(C)C(=O)[C@@H](NCCOc2ccc(F)cc2CCCNC(=O)[C@@H](Cc2ccc(F)cc2)NC1=O)C1CC1
    Show/Hide
Compound Formula C29H36F2N4O4
Compound Structure
Protein Name
 Protein Info 
Growth hormone secretagogue receptor type 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
GRP-related receptor
Uniprot ID
Q92847
Gene Name
GHSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
Ki = 10 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 58 nM