Brief Information of the Compound and Protein
Compound Name
N-(4-Chloro-3-((1-nicotinoylpiperidin-4-yl)oxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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PubChem ID
CID: 134150061
Canonical SMILES
CN1CCN(Cc2ccc(C(=O)Nc3ccc(Cl)c(OC4CCN(C(=O)c5cccnc5)CC4)c3)cc2C(F)(F)F)CC1
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Compound Formula C31H33ClF3N5O3
Compound Structure
Protein Name
Mast/stem cell growth factor receptor Kit
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
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TK protein kinase group
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Tyrosine protein kinase PDGFR family
Uniprot ID
P10721
Gene Name
KIT
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
GI50 = 340 nM
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