Brief Information of the Compound and Protein
Compound Name
2-fluoro-4-[5-[2-(4-methyl-1-oxo-3H-2-benzofuran-5-yl)ethyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]benzonitrile
    Show/Hide
PubChem ID
CID: 91810383
Canonical SMILES
Cc1c2COC(=O)c2ccc1CCN1CCc2c(C1)cnn2-c1ccc(C#N)c(F)c1
    Show/Hide
Compound Formula C24H21FN4O2
Compound Structure
Protein Name
ATP-sensitive inward rectifier potassium channel 1
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Potassium channels
>
Inwardly rectifying potassium channel
Uniprot ID
P48048
Gene Name
KCNJ1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 27.46 nM
   TI
   LI
   LO
   TS