Brief Information of the Compound and Protein
Compound Name
US9012443, 12
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PubChem ID
CID: 71585930
SID: 163638115
Canonical SMILES
COc1cc(ccc1-c1cccc2cc(ccc12)S(=O)(=O)Nc1ncns1)C(F)(F)F
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Compound Formula C20H14F3N3O3S2
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
>
Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
IC50 = 11600 nM
   TI
   LI
   LO
   TS
2
IC50 = 12000 nM
   TI
   LI
   LO
   TS