Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-(1H-indazol-5-yl)-N-methyl-4-pyridin-2-yl-1,3-thiazol-2-amine
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 PubChem ID
CID: 127052038
Canonical SMILES
CN(c1nc(cs1)-c1ccccn1)c1ccc2[nH]ncc2c1
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Compound Formula C16H13N5S
Compound Structure
Protein Name
 Protein Info 
Glutamate receptor 1
Protein Classification
Ion channel
>
Ligand-gated ion channel
>
Ionotropic glutamate receptor
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AMPA receptor
Uniprot ID
P42261
Gene Name
GRIA1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000470 CHO-S
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 147 nM
   TI
   LI
   LO
   TS
2
IC50 > 83300 nM
   TI
   LI
   LO
   TS