Brief Information of the Compound and Protein
Compound Name
N-methyl-N-(1-pyridin-2-ylpyrazol-3-yl)-1H-indazol-5-amine
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PubChem ID
CID: 127052039
Canonical SMILES
CN(c1ccn(n1)-c1ccccn1)c1ccc2[nH]ncc2c1
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Compound Formula C16H14N6
Compound Structure
Protein Name
Glutamate receptor 1
Protein Classification
Ion channel
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Ligand-gated ion channel
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Ionotropic glutamate receptor
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AMPA receptor
Uniprot ID
P42261
Gene Name
GRIA1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000470 CHO-S Cricetulus griseus (Chinese hamster)  2
1
IC50 = 353 nM
   TI
   LI
   LO
   TS
2
IC50 > 83300 nM
   TI
   LI
   LO
   TS