Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(4R)-6-(3-cyclopropyl-1-methylindazol-5-yl)-4-methyl-1,3,4,5-tetrahydro-1,5-benzodiazepin-2-one
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 PubChem ID
CID: 121271781
Canonical SMILES
C[C@@H]1CC(=O)Nc2cccc(-c3ccc4n(C)nc(C5CC5)c4c3)c2N1
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Compound Formula C21H22N4O
Compound Structure
Protein Name
 Protein Info 
CREB-binding protein
Protein Classification
Epigenetic regulator
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Bromodomain
Uniprot ID
Q92793
Gene Name
CREBBP
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 3000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 33 nM