Brief Information of the Compound and Protein
Compound Name
2-[[3-(2,6-dichlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-6-[4-(trifluoromethoxy)phenyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
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PubChem ID
CID: 58044619
Canonical SMILES
FC(F)(F)Oc1ccc(cc1)-c1ccc2nn(Cc3nc(no3)-c3c(Cl)cccc3Cl)c(=O)n2c1
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Compound Formula C22H12Cl2F3N5O3
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 3500 nM
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