Brief Information of the Compound and Protein
Compound Name
2-N-(2,6-dimethylphenyl)-3-methyl-4-N,4-N-dipropylbenzimidazole-2,4-diamine;2,2,2-trifluoroacetic acid
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PubChem ID
CID: 127030336
Canonical SMILES
OC(=O)C(F)(F)F.CCCN(CCC)c1cccc2nc(Nc3c(C)cccc3C)n(C)c12
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Compound Formula C24H31F3N4O2
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 140 nM
   TI
   LI
   LO
   TS