Brief Information of the Compound and Protein
Compound Name
(5R*)-N5-(5-Bromothiazol-2-yl)-(6R*)-N6-(3-(4-methyl piperazin-1-yl)-propyl)-(4S*,7R*)-[4,7-ethenylene-spiro[2.4]heptane]-5,6-dicarboxamide
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PubChem ID
CID: 87422158
Canonical SMILES
CN1CCN(CCCNC(=O)[C@H]2[C@H](C(=O)Nc3ncc(Br)s3)[C@@H]3C=C[C@H]2C32CC2)CC1
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Compound Formula C22H30BrN5O2S
Compound Structure
Protein Name
N-formyl peptide receptor 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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N-formyl methionyl peptide receptor
Uniprot ID
P25090
Gene Name
FPR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 49 nM
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