Brief Information of the Compound and Protein
Compound Name
(5R*)-N5-(4-Acetyl-thiazol-2-yl-methyl)-(6R*)-N6-(3-(1H-benzoimidazol-2-yl)-propyl)-(4S*,7R*)-[4,7-ethenylene-spiro[2.4]heptane]-5,6-dicarboxamide
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PubChem ID
CID: 67495041
Canonical SMILES
CC(=O)c1csc(CNC(=O)[C@H]2[C@H](C(=O)NCCCc3nc4ccccc4[nH]3)[C@H]3C=C[C@@H]2C32CC2)n1
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Compound Formula C27H29N5O3S
Compound Structure
Protein Name
N-formyl peptide receptor 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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N-formyl methionyl peptide receptor
Uniprot ID
P25090
Gene Name
FPR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 106 nM
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